Molecule Details
InChIKeyYGQJBWJOHRVWHU-UHFFFAOYSA-N
Compound Name4-[[1-[3-[(4-Bromobenzoyl)amino]phenyl]-3-(dimethylamino)propyl]amino]quinazoline-8-carboxamide
Canonical SMILESCN(C)CCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)c2ccc(Br)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.9 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 8.3 IC50 ChEMBL;BindingDB