Molecule Details
InChIKeyYFOHBZPJQXLDMO-UHFFFAOYSA-N
Compound Name1,3-dimethyl-6-[4-[2-oxo-2-(4-phenylpiperazin-1-yl)ethoxy]phenyl]-5H-pyrrolo[3,2-d]pyrimidine-2,4-dione
Canonical SMILESCn1c(=O)c2[nH]c(-c3ccc(OCC(=O)N4CCN(c5ccccc5)CC4)cc3)cc2n(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB