Molecule Details
InChIKeyYFBAOXITVIDIPH-UHFFFAOYSA-N
Compound Name1-[3-[(4,4-Dimethyl-8-morpholin-4-yl-11-thia-9,14,16-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-1,7,9,12,14,16-hexaen-13-yl)amino]propyl]pyrrolidin-2-one
Canonical SMILESCC1(C)CCc2c(N3CCOCC3)nc3sc4c(NCCCN5CCCC5=O)ncnc4c3c2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27815 PDE4A Homo sapiens Human PF18100 PF00233 7.7 IC50 ChEMBL;BindingDB
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 7.7 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 7.2 IC50 ChEMBL;BindingDB