Molecule Details
InChIKeyYEXGHTGVNJDCFJ-UHFFFAOYSA-N
Compound Name4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino]-N-[2-(2,4-dichloro-phenyl)-ethyl]-benzamide
Canonical SMILESO=C(NCCc1ccc(Cl)cc1Cl)c1ccc(N/C(=N/C2CCCCC2)N2CCNCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33032 MC5R Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB