Molecule Details
InChIKeyYESKHRZGFKDGEH-UHFFFAOYSA-N
Compound Name8,8-difluoro-N-[5-[2-(1-methylpyrazol-4-yl)pyridin-4-yl]oxypyridin-2-yl]-1-oxo-2-azaspiro[4.4]nonane-2-carboxamide
Canonical SMILESCn1cc(-c2cc(Oc3ccc(NC(=O)N4CCC5(CCC(F)(F)C5)C4=O)nc3)ccn2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 8.6 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 8.0 IC50 ChEMBL;BindingDB
P16234 PDGFRA Homo sapiens Human PF07679 PF25305 PF07714 7.4 IC50 ChEMBL;BindingDB