Molecule Details
InChIKeyYERMBKYNILMCNC-VQTJNVASSA-N
Compound Nametrans-(1R,2R)-N-[4-(benzenesulfonyl)phenyl]-2-pyridin-3-ylcyclopropane-1-carboxamide
Canonical SMILESO=C(Nc1ccc(S(=O)(=O)c2ccccc2)cc1)[C@@H]1C[C@H]1c1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 7.0 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB
P43490 NAMPT Homo sapiens Human PF18127 PF04095 6.0 IC50 ChEMBL;BindingDB