Molecule Details
InChIKeyYENLCWWOFXIPIH-QOAPGFADSA-N
Compound Name(S)-2-{(S)-3-Carboxy-2-[(2S,5S)-5-[3-(1-ethyl-propyl)-ureido]-6,6-dimethyl-4-oxo-2-(2-oxo-2-pyrrolidin-1-yl-ethyl)-heptanoylamino]-propionylamino}-4-methyl-pentanoic acid
Canonical SMILESCCC(CC)NC(=O)N[C@H](C(=O)C[C@@H](CC(=O)N1CCCC1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)O)C(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23921 RRM1 Homo sapiens Human PF03477 PF02867 PF00317 8.2 IC50 ChEMBL;BindingDB
P31350 RRM2 Homo sapiens Human PF00268 8.2 IC50 ChEMBL
Q7LG56 RRM2B Homo sapiens Human PF00268 8.2 IC50 ChEMBL