Molecule Details
InChIKeyYEGXHTKFBQFSNF-UHFFFAOYSA-N
Compound Name1-(1-Azabicyclo[2.2.2]octan-3-yl)-3,4-dichloro-2-iodopyrrolo[2,3-b]pyridine-6-carboxamide
Canonical SMILESNC(=O)c1cc(Cl)c2c(Cl)c(I)n(C3CN4CCC3CC4)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB