Molecule Details
InChIKeyYDXHIJKYXAXQTE-UHFFFAOYSA-N
Canonical SMILESCC1(C)CC(C(Nc2cnc(-n3cc(C(F)(F)F)cn3)nc2)c2ccc(C(=O)NCCC(=O)O)cc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P01275 GCG Homo sapiens Human PF00123 8.3 Ki ChEMBL;BindingDB
P47871 GCGR Homo sapiens Human PF00002 PF02793 8.2 Ki ChEMBL;BindingDB