Molecule Details
InChIKeyYDQQLXXIRZYPPK-CGXNFDGLSA-N
Compound Name(R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propylamino)-3-methyl-butyryl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-hexanoic acid
Canonical SMILESCCCC[C@@H](NC(=O)[C@@H]1Cc2ccccc2CN1C(=O)[C@@H](NC[C@@H](N)CS)C(C)C)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.9 pIC50 TTD_MultiTarget
P53609 PGGT1B Homo sapiens Human PF00432 8.9 IC50 ChEMBL
P49356 FNTB Homo sapiens Human PF00432 6.1 IC50 ChEMBL;BindingDB