Molecule Details
InChIKeyYDAHPXSXJZMUPN-UHFFFAOYSA-N
Canonical SMILESCCc1nc2c(C)cc(C)nc2n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)C(c2ccccc2)c2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 10.3 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 7.7 IC50 ChEMBL;BindingDB