Molecule Details
InChIKeyYCZXNWIFFVKUST-UHFFFAOYSA-N
Compound Name5-chloro-N-[6-[2-(methylamino)propanoylamino]-4-(1,3,5-trimethylpyrazolo[4,5-d]pyrimidin-7-yl)-2-pyridinyl]pyridine-2-carboxamide
Canonical SMILESCNC(C)C(=O)Nc1cc(-c2nc(C)nc3c(C)nn(C)c23)cc(NC(=O)c2ccc(Cl)cn2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.24
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P98170 XIAP Homo sapiens Human PF00653 PF21290 PF13920 8.2 IC50 ChEMBL;BindingDB
Q13489 BIRC3 Homo sapiens Human PF00653 PF00619 PF21290 PF13920 8.2 IC50 BindingDB
Q13490 BIRC2 Homo sapiens Human PF00653 PF00619 PF21290 PF13920 8.2 IC50 ChEMBL