Molecule Details
InChIKeyYCWMLVXTEBFVHL-HXUWFJFHSA-N
Compound Name6,7-dimethoxy-4-[(3R)-3-[(7-methoxynaphthalen-2-yl)oxy]pyrrolidin-1-yl]quinazoline
Canonical SMILESCOc1ccc2ccc(O[C@@H]3CCN(c4ncnc5cc(OC)c(OC)cc45)C3)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 7.8 Ki ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.6 Ki ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.5 Ki ChEMBL;BindingDB