Molecule Details
InChIKeyYCLIWTLPTXAGPQ-UHFFFAOYSA-N
Compound Name4-[(3,5-Dichloro-4-Methoxyphenyl)amino]-6-Methoxy-7-[3-(4-Methylpiperazin-1-Yl)propoxy]quinoline-3-Carbonitrile
Canonical SMILESCOc1cc2c(Nc3cc(Cl)c(OC)c(Cl)c3)c(C#N)cnc2cc1OCCCN1CCN(C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0C1S8 WEE2 Homo sapiens Human PF00069 8.3 Kd ChEMBL;BindingDB
P30291 WEE1 Homo sapiens Human PF00069 7.4 Kd ChEMBL;BindingDB
Q99640 PKMYT1 Homo sapiens Human PF00069 6.3 Kd ChEMBL;BindingDB