Molecule Details
InChIKeyYCHHLNUILPSKGG-UHFFFAOYSA-N
Compound Name3-[4-(1-cyclopropylpyrazol-4-yl)-3-pyridinyl]-N-[4-(morpholin-4-ylmethyl)phenyl]propanamide
Canonical SMILESO=C(CCc1cnccc1-c1cnn(C2CC2)c1)Nc1ccc(CN2CCOCC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 7.5 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 7.5 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB