Molecule Details
InChIKeyYBFJEMNJNCMXOO-UHFFFAOYSA-N
Compound Name1-[1-[1-(2-hydroxyethyl)-6-oxo-3-pyridinyl]-3-propan-2-ylpyrazol-5-yl]-3-[4-[6-(1H-indazol-5-ylamino)pyrimidin-4-yl]oxynaphthalen-1-yl]urea
Canonical SMILESCC(C)c1cc(NC(=O)Nc2ccc(Oc3cc(Nc4ccc5[nH]ncc5c4)ncn3)c3ccccc23)n(-c2ccc(=O)n(CCO)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.5 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.9 IC50 ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB