Molecule Details
InChIKeyYARZXKRRRMSSKW-UHFFFAOYSA-N
Compound Name3-[3-(4-Acetoxy-4-phenyl-piperidin-1-yl)-propylcarbamoyl]-4-(3,4-difluoro-phenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester
Canonical SMILESCOC(=O)C1=C(C)NC(=O)N(C(=O)NCCCN2CCC(OC(C)=O)(c3ccccc3)CC2)C1c1ccc(F)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB