Molecule Details
InChIKeyYAQRTUXYVQSHDL-UHFFFAOYSA-N
Compound Name1',2'-dibenzyl-5'-ethylspiro[1,2-dihydroindene-3,7'-8H-imidazo[2,1-b]purine]-4'-one
Canonical SMILESCCN1C(=O)c2nc(Cc3ccccc3)n(Cc3ccccc3)c2N2CC3(CCc4ccccc43)N=C12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HCR9 PDE11A Homo sapiens Human PF01590 PF00233 6.8 IC50 ChEMBL;BindingDB
Q99572 P2RX7 Homo sapiens Human PF20478 PF00864 6.6 IC50 ChEMBL;BindingDB