Molecule Details
InChIKeyYANNSWWYRMATEM-JTQLQIEISA-N
Compound Name8-bromo-2-{[(3S)-3-(methyloxy)pyrrolidin-1-yl]methyl}[1]benzofuro[3,2-d]pyrimidin-4(3H)-one
Canonical SMILESCO[C@H]1CCN(Cc2nc3c(oc4ccc(Br)cc43)c(=O)[nH]2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL6.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P67870 CSNK2B Homo sapiens Human PF01214 6.3 IC50 ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 6.3 IC50 ChEMBL