Molecule Details
InChIKeyYACUPCZEGXPESB-UHFFFAOYSA-N
Compound Name4-(2-Hydroxy-ethyl)-N-[2-(N-methyl-guanidino)-acetyl]-benzenesulfonamide
Canonical SMILESCN(CC(=O)NS(=O)(=O)c1ccc(CCO)cc1)C(=N)N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.93
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.4 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.4 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.0 Ki ChEMBL;BindingDB