Molecule Details
InChIKeyXZPYWTFDULVLJE-UHFFFAOYSA-N
Compound Name2-(4-tert-butylphenyl)-N-[1-[(5-cyano-2-pyridinyl)methyl]pyrazol-3-yl]acetamide
Canonical SMILESCC(C)(C)c1ccc(CC(=O)Nc2ccn(Cc3ccc(C#N)cn3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.6 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 8.6 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 8.1 IC50 ChEMBL;BindingDB