Molecule Details
InChIKeyXZEVSGANERUOOE-UHFFFAOYSA-N
Compound NameTert-butyl 5-[2-[1-(6-carbamoylthieno[3,2-d]pyrimidin-4-yl)piperidin-4-yl]ethylcarbamoyl]thiophene-2-carboxylate
Canonical SMILESCC(C)(C)OC(=O)c1ccc(C(=O)NCCC2CCN(c3ncnc4cc(C(N)=O)sc34)CC2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8IXJ6 SIRT2 Homo sapiens Human PF02146 8.7 IC50 ChEMBL;BindingDB
Q9NTG7 SIRT3 Homo sapiens Human PF02146 8.5 IC50 ChEMBL;BindingDB
Q96EB6 SIRT1 Homo sapiens Human PF02146 8.2 IC50 ChEMBL;BindingDB