Molecule Details
InChIKeyXYZNJJAFIUQYLC-UHFFFAOYSA-N
Compound Name4-(4-(1,2-dimethyl-1H-imidazol-5-yl)pyrimidin-2-ylamino)-N-(2-methoxyethyl)benzenesulfonamide
Canonical SMILESCOCCN[S@SP3](=O)(=O)c1ccc(Nc2nccc(-c3cnc(C)n3C)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.1
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.1 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.1 pIC50 TTD_MultiTarget