Molecule Details
InChIKeyXYMYMSOAMWEUBS-UHFFFAOYSA-N
Compound NameIndolo[6,7-a]pyrrolo[3,4-c]carbazole deriv. 3e
Canonical SMILESCn1ccc2ccc3c4[nH]c5cccc(Br)c5c4c4c(c3c21)C(=O)NC4=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 6.9 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.9 pIC50 TTD_MultiTarget
P24385 CCND1 Homo sapiens Human PF02984 PF00134 6.8 IC50 ChEMBL