Molecule Details
InChIKeyXXTLQVLGJWHTST-UHFFFAOYSA-N
Compound Name6-[6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridin-1-yl]-N-piperidin-4-ylpyridin-2-amine
Canonical SMILESCc1cncc(-c2cc3c(cn2)cnn3-c2cccc(NC3CCNCC3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.6 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.9 Ki ChEMBL;BindingDB