Molecule Details
InChIKeyXWJOKKXDMHSILW-UHFFFAOYSA-N
Compound NameN-Benzyl-3-({[5-(Pyridin-4-Yl)-4h-1,2,4-Triazol-3-Yl]methyl}amino)benzamide
Canonical SMILESO=C(NCc1ccccc1)c1cccc(NCc2nc(-c3ccncc3)n[nH]2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35626 GRK3 Homo sapiens Human PF00169 PF00069 PF00615 8.7 IC50 ChEMBL;BindingDB
P25098 GRK2 Homo sapiens Human PF00169 PF00069 PF00615 8.2 IC50 ChEMBL;BindingDB
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 7.6 IC50 ChEMBL;BindingDB