Molecule Details
InChIKeyXVYMHUPUYXWRAO-UHFFFAOYSA-N
Compound Name(1-{1-Benzyl-2-oxo-2-[3-(3,4,4a,8a-tetrahydro-1H-isoquinolin-2-yl)-propylcarbamoyl]-ethylcarbamoyl}-3-methyl-butyl)-carbamic acid benzyl ester
Canonical SMILESCC(C)CC(NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(=O)C(=O)NCCCN1CCC2C=CC=CC2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.24
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P17655 CAPN2 Homo sapiens Human PF01067 PF13833 PF00648 9.7 Ki BindingDB
P07384 CAPN1 Homo sapiens Human PF01067 PF13833 PF00648 9.7 Ki BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 8.3 Ki BindingDB