Molecule Details
InChIKeyXVWWDCXPGPSOQP-UHFFFAOYSA-N
Compound Name6-[2-(1-Cyclohexyl-2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-yl)-cyclopropyl]-naphthalene-2-carboxamidine
Canonical SMILESCN1CCc2ccc(C3CC3c3ccc4cc(C(=N)N)ccc4c3)cc2C1C1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00749 PLAU Homo sapiens Human PF00051 PF00089 7.5 Ki ChEMBL;BindingDB
P06870 KLK1 Homo sapiens Human PF00089 6.5 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 6.1 Ki ChEMBL;BindingDB