Molecule Details
InChIKeyXVKWLASBXAWEPG-CQSZACIVSA-N
Compound Name(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidin-2-yl)((R)-2-(methoxymethyl)pyrrolidin-1-yl)methanone
Canonical SMILESCOC[C@H]1CCCN1C(=O)c1cn2c(-c3ccc(Cl)cc3Cl)c(CN)c(C)nc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 8.9 Ki ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 8.9 Ki ChEMBL;BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 8.5 Ki ChEMBL;BindingDB