Molecule Details
InChIKeyXVGGLWKPTSTHJU-UHFFFAOYSA-N
Compound NameN,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine
Canonical SMILESCCN(CC)CCCOc1ccc2c(c1)CN(C)CC2c1ccc(OC)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5N1 HRH3 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.4 Ki ChEMBL;BindingDB