Molecule Details
InChIKeyXUVYYIIVCVDGFW-XZOQPEGZSA-N
Canonical SMILESO=C(N[C@H]1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)[C@H](Cc2ccccc2)C1)c1cc(O)nc2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P29371 TACR3 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB