Molecule Details
InChIKeyXULJUQRQXLWPOJ-LWQYYNMXSA-N
Compound Name2-[3-(butanoylamino)-5-[(2S,4R)-6-carbamimidoyl-4-methyl-4-phenyl-2,3-dihydro-1H-quinolin-2-yl]phenyl]-5-carbamoylbenzoic acid
Canonical SMILESCCCC(=O)Nc1cc(-c2ccc(C(N)=O)cc2C(=O)O)cc([C@@H]2C[C@](C)(c3ccccc3)c3cc(C(=N)N)ccc3N2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 9.5 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.3 Ki ChEMBL
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.2 Ki ChEMBL;BindingDB