Molecule Details
InChIKeyXUJJWQQLMFLJKO-SQHAQQRYSA-N
Compound Name3'-Amino-5'-[(2s,4r)-6-Carbamimidoyl-4-Phenyl-1,2,3,4-Tetrahydroquinolin-2-Yl]biphenyl-2-Carboxylic Acid
Canonical SMILESN=C(N)c1ccc2c(c1)[C@@H](c1ccccc1)C[C@@H](c1cc(N)cc(-c3ccccc3C(=O)O)c1)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 8.1 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.4 Ki ChEMBL
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.2 Ki ChEMBL;BindingDB