Molecule Details
InChIKeyXTWXMJDVQOEURD-SOFGYWHQSA-N
Compound Name4-methyl-3-(3-((4-methylpiperazin-1-yl)methyl)styryl)-1H-indazole-5-carbonitrile
Canonical SMILESCc1c(C#N)ccc2[nH]nc(/C=C/c3cccc(CN4CCN(C)CC4)c3)c12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.78
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget