Molecule Details
InChIKeyXTPTVAPEXHUUDR-UHFFFAOYSA-N
Compound Name4-(Piperazin-1-yl)-2,6-di(pyrrolidin-1-yl)pyrimidine
Canonical SMILESc1c(N2CCCC2)nc(N2CCCC2)nc1N1CCNCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P51878 CASP5 Homo sapiens Human PF00619 PF00656 7.0 IC50 ChEMBL;BindingDB
P29466 CASP1 Homo sapiens Human PF00619 PF00656 6.6 IC50 ChEMBL;BindingDB
P49662 CASP4 Homo sapiens Human PF00619 PF00656 6.5 IC50 ChEMBL;BindingDB