Molecule Details
InChIKeyXTKSMYZRQMTSMS-UHFFFAOYSA-N
Compound Name3-(5-{[(3-Oxo-3,4-dihydroquinoxalin-2-YL)methyl]sulfanyl}-1,3,4-thiadiazol-2-YL)-1-[3-(trifluoromethyl)phenyl]urea
Canonical SMILESO=C(Nc1cccc(C(F)(F)F)c1)Nc1nnc(SCc2nc3ccccc3[nH]c2=O)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.1 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 8.1 IC50 ChEMBL
P04629 NTRK1 Homo sapiens Human PF13855 PF16920 PF07714 PF18613 6.6 IC50 ChEMBL;BindingDB