Molecule Details
InChIKeyXTDBGBVPMKZZHK-UHFFFAOYSA-N
Compound Name2-[3-[(7-Cyclohexylpyrrolo[2,3-d]pyrimidin-2-yl)amino]phenyl]acetic acid
Canonical SMILESO=C(O)Cc1cccc(Nc2ncc3ccn(C4CCCCC4)c3n2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.22
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.2 IC50 ChEMBL
P11802 CDK4 Homo sapiens Human PF00069 9.2 pIC50 TTD_MultiTarget