Molecule Details
InChIKeyXTASITJXTTXPJS-UHFFFAOYSA-N
Compound NameUS9732063, Example 2
Canonical SMILESCOc1ccc(-n2nc(C(C)(C)C)cc2NC(=O)Nc2ccc(Oc3ccnc(Nc4cccc(N=S(C)(C)=O)c4)n3)c3ccccc23)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.1 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.8 IC50 ChEMBL;BindingDB
P53778 MAPK12 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB