Target not found.
Molecule Details
InChIKeyXSJWROYTYXTZKU-UHFFFAOYSA-N
Compound Name2-(1H-pyrazol-4-yl)-N-[4-(pyrazol-1-ylmethyl)phenyl]-1H-pyrrolo[3,2-c]pyridin-6-amine
Canonical SMILESc1cnn(Cc2ccc(Nc3cc4[nH]c(-c5cn[nH]c5)cc4cn3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P20248 CCNA2 Homo sapiens Human PF02984 PF00134 PF16500 7.6 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB