Molecule Details
InChIKeyXSJMSGALWUODPK-UHFFFAOYSA-N
Compound NameSdccggsk-0000152.P001
Canonical SMILESCOc1cc(Nc2nccc(-c3cnn4ncccc34)n2)cc(OC)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget
P49841 GSK3B Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB