Molecule Details
InChIKeyXSHSZTXMXLVUME-INIZCTEOSA-N
Compound Name4-Amino-6,7-dimethoxy-2-[(3S)-3-(t-butylcarbamoyl)-4-(2-furoyl)-1-piperazinyl]-quinazoline
Canonical SMILESCOc1cc2nc(N3CCN(C(=O)c4ccco4)[C@H](C(=O)NC(C)(C)C)C3)nc(N)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35368 ADRA1B Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB