Molecule Details
InChIKeyXRRMKGIMNWBQJX-UHFFFAOYSA-N
Compound Name3-(2-cyclopentylacetyl)-6-ethyl-1H-quinolin-4-one
Canonical SMILESCCc1ccc2[nH]cc(C(=O)CC3CCCC3)c(=O)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14867 GABRA1 Homo sapiens Human PF02931 PF02932 8.3 Ki ChEMBL;BindingDB
P18507 GABRG2 Homo sapiens Human PF02931 PF02932 8.3 Ki ChEMBL
P47870 GABRB2 Homo sapiens Human PF02931 PF02932 8.3 Ki ChEMBL