Molecule Details
InChIKeyXREDUPOVEQDQQS-UHFFFAOYSA-N
Compound NameDiamino-5-phenyl-6-ethylpyrimidine, 2,4-
Canonical SMILESCCc1nc(N)nc(N)c1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.15
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07577
Drug Name2,4-Diamino-5-phenyl-6-ethylpyrimidine
CAS Number27653-49-2
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 18788 CHEMBL22148 ChemSpider: 84060 PDB: CP7 PubChem:93114 PubChem:99444048 ZINC: ZINC000013282257
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 8.0 Ki ChEMBL;BindingDB
O02604 Plasmodium vivax Pathogen PF00186 PF00303 10.3 Ki BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P04818 TYMS Thymidylate synthase binder targets
P12461 P12461 Thymidylate synthase inhibitor targets