Molecule Details
InChIKeyXQOMHPQXEDJCGI-JDBXKHNRSA-N
Compound NameH-D-Phe-D-Cys(1)-Phe-N(Me)Trp-Lys-Thr-Cys(1)-Thr-NH2
Canonical SMILESC[C@@H](O)[C@H](NC(=O)[C@@H]1CSSC[C@@H](NC(=O)[C@H](N)Cc2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N1)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35346 SSTR5 Homo sapiens Human PF00001 9.2 Kd ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 8.0 Kd ChEMBL;BindingDB
P30874 SSTR2 Homo sapiens Human PF00001 7.6 Kd ChEMBL;BindingDB