Molecule Details
InChIKeyXQNDLDMSQNGBNX-VABKMULXSA-N
Canonical SMILESCOC[C@@H]1C[C@H](OC)CN1Cc1ncc(-c2cccc(-c3cccc(-c4cnc(CNC[C@@H]5CCC(=O)N5)c(OC)n4)c3Cl)c2Cl)nc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15116 PDCD1 Homo sapiens Human PF07686 9.7 IC50 ChEMBL;BindingDB
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 9.7 IC50 ChEMBL