Molecule Details
InChIKeyXQEZXMGUDOPHOF-UHFFFAOYSA-N
Compound Name1-[(8-Bromo-4-oxo-3,4-dihydro[1]benzofuro[3,2-d]pyrimidin-2-yl)methyl]pyrrolidine-3-carboxylic acid
Canonical SMILESO=C(O)C1CCN(Cc2nc3c(oc4ccc(Br)cc43)c(=O)[nH]2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P67870 CSNK2B Homo sapiens Human PF01214 7.3 IC50 ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 7.3 IC50 ChEMBL
P11309 PIM1 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB