Molecule Details
InChIKeyXPRDGKCNHYYXEJ-UHFFFAOYSA-N
Canonical SMILESCc1cc(C)n2nc(CC3=C(O)CC(CCc4ccc(C(C)(C)C#N)c(F)c4)(C4CCCC4)OC3=O)nc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.52
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10635 CYP2D6 Homo sapiens Human PF00067 6.5 IC50 ChEMBL
Q8JXU8 NS5B Hepacivirus hominis Pathogen PF00998 8.5 IC50 ChEMBL