Molecule Details
InChIKeyXOVJPFAQAXPONH-UHFFFAOYSA-N
Compound NamePyrazolo[3,4-d]pyrimidin-4-one deriv. 19e
Canonical SMILESCCc1nn(-c2c(Cl)cc(Cl)cc2Cl)c2nc(Cc3cccc(C)c3)[nH]c(=O)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
O96020 CCNE2 Homo sapiens Human PF02984 PF00134 6.4 IC50 ChEMBL
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 6.4 IC50 ChEMBL