Molecule Details
InChIKeyXOFGTUXJGBWWCZ-UHFFFAOYSA-N
Canonical SMILESO=C(O)CC1CCC2(CC1)CCN(c1ccc(NC(=O)c3nnc(Nc4ccc(F)c(F)c4)o3)cn1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.58
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75907 DGAT1 Homo sapiens Human PF03062 7.8 IC50 ChEMBL
P24752 ACAT1 Homo sapiens Human PF02803 PF00108 7.3 IC50 ChEMBL