Molecule Details
InChIKeyXOFBXIHLMNJMOE-UHFFFAOYSA-N
Compound Name15,20-Dioxo-2-oxa-9,11,16,19-tetrazapentacyclo[19.6.2.13,7.09,13.025,29]triaconta-1(28),3,5,7(30),10,12,21,23,25(29),26-decaene-4-carbonitrile
Canonical SMILESN#Cc1ccc2cc1Oc1ccc3cccc(c3c1)C(=O)NCCNC(=O)Cc1cncn1C2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.93
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.6 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.6 IC50 ChEMBL